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API | Intermediates | Cas No. |
---|---|---|
Apalutamide | 5-Amino-3-(Trifluoromethyl)-Picolinonitrile | 573762-62-6 |
Asenapine | Trans-11-Chloro-2,3,3a,12b-Tetrahydro-2-Methyl-1h-Dibenz[2,3:6,7]Oxepino[4,5-C]Pyrrol-1-One | 129385-59-7 |
Atogepant | Tert-Butyl((3s,5s,6r)-6-Methyl-2-Oxo-5-(2,3,6-Trifluorophenyl)Piperidin-3-Yl)Carbamate | 1456803-43-2 |
Aliskiren | Trans-1,4-Dichloro-2-butene | 110-57-6 |
Avatrombopag | 4-(4-Chlorothiophen-2-Yl)Thiazol-2-Amine | 570407-10-2 |
Bicalutamide | 4-Amino-3-(Trifluoromethyl)Benzonitrile | 654-70-6 |
Carfilzomib | (S)-2-Amino-4-Methyl-1-((R)-2-Methyloxiran-2-yl)pentan-1-one, trifluoroacetate | 247068-85-5 |
Dabrafenib | Methyl 3-(2,6-Difluorophenylsulfonamido)-2-Fluorobenzoate | 1195768-19-4 |
3-Amino-2-Fluorobenzoic Acid Methyl Ester | 1195768-18-3 | |
Dapagliflozin | (2R,3R,4R,5S,6S)-2-(Acetoxymethyl)-6-(4-chloro-3-(4-ethoxybenzyl)phenyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate | 461432-25-7 |
Darunavir | (3R,3aS,6aR)-Carbonic Acid 2,5-Dioxopyrrolidin-1-yl Ester Hexahydrofur[2,3-b]Furan-3-yl Ester | 799241-85-3 |
Deflazacort | (11b,16b)-11-Hydroxy-2-Methyl-5H-Pregna-1,4-Dieno(17,16-D)Oxazole-3,20-Dione(D-5) | 13649-88-2 |
Dolutegravir | Methyl 4-Methoxyacetoacetate | 41051-15-4 |
2,4-Difluorobenzylamine | 455-13-0 | |
Dolasetron | Aminoacetaldehyde Dimethyl Acetal | 22483-09-6 |
Docetaxel | (4S,5R)-2-(4-Methoxyphenyl)-N-t-Boc-4-Phenyl-Oxazolidine-5-Carboxylic Acid | 196404-55-4 |
Eltrombopag | 3-Amino-2-Hydroxybenzo[h]-3-Carboxylic Acid | 376592-93-7 |
Empagliflozin | (1S)-1,5-Anhydro-1-C-[4-Chloro-3-[[4-[[(3S)-Tetrahydro-3- Furanyl]oxy]phenyl]methyl]phenyl]-D-Glucitol Tetraacetate | 915095-99-7 |
Ezetimibe | S(+)4-Phenyl-2-Oxazolidinone (SPOZ) | 99395-88-7 |
Finerenone | 2-Cyanoethylacetoacetate | 65193-87-5 |
4-Amino-5-Methylpyridin-2-ol; 4-Amino-2-hydroxy-5-methylpyridine | 95306-64-2 | |
4-Cyano-2-Methoxybenzaldehyde | 21962-45-8 | |
(Z)-2-Cyanoethyl-2-(4-Cyano-2-Methoxybenzylidene)-3-Oxobutanoate | 1050477-39-8 | |
Finasteride | N-Tert-Butyl-3-Oxo-4-Aza-5a-Androst-17b-Carboxamide | 166896-74-8 |
Fulvestrant | (7a,17b)-7-(9-Bromononyl)-estra-1,3,5(10)-triene-3,17-diol-17-acetateN-3 | 875573-66-3 |
(7a,17b)-7-[9-([4,4,5,5,5-Pentafluoropentyl]thio)nonyl]-estra-1,3,5(10)-triene-3,17-diol N-1 | 153004-31-0 | |
(7a,17b)-7-[9-[4,4,5,5,5-Pentafluoropentyl] Sulfinyl[Nonyl]Estra-1,3,5-(10)-Triene-3-Diol-17-Oxyethyl | 875573-69-6 | |
4,4,5,5,5-Pentafluoro-1-pentanol | 148043-73-6 | |
Gliclazide | 3-Amino-3-azabicyclo[3.3.0]octane hydrochloride | 58108-05-7 |
Irinotecan | 7-Ethyl-10-hydroxycamptothecin | 86639-52-3 |
1-Chlorocarbonyl-4-piperidinopiperidine hydrochloride | 143254-82-4 | |
Isavuconazole | (2R,3R)-3-(2,5-Difluorophenyl)-3-Hydroxy-2-Methyl-4-(1H-1,2,4-Triazol-1-yl)Thiobutyramide | 368421-58-3 |
(2-(Methylamino) Pyridin-3-yl) Methyl 2-(Tert-Butoxycarbonyl)(Methyl)Amino) Acetate | 1180002-01-0 | |
Glycine,N-[(1,1-dimethylethoxy)carbonyl]-N-Methyl-, [2-[[[(1-chloroethoxy)carbonyl]Methylamino]-3-pyridinyl]Methyl]ester | 338990-31-1 | |
2-(Methylamino)pyridine-3-methanol | 32399-12-5 | |
4-Cyanophenacyl Bromide | 20099-89-2 | |
Ketoprofen | 3-(1-Cyanoethyl)Benzoic Acid/CEВА | 5537-71-3 |
Ketoprofen Nitrile | 42872-30-0 | |
Lifitegrast | 6-Isoquinolinecarboxylic Acid, 5,7-Dichloro-1,2,3,4-Tetrahydro, Hydrochloride | 1289646-93-0 |
(S)-methyl 2-amino-3-(3-(methylsulfonyl)phenyl)propanoate hydrochloride | 851785-21-2 | |
Benzofuran-6-Carboxylic Acid | 77095-51-3 | |
Lorbrena | Tert-Butyl N-[(4-Bromo-5-Cyano-1-Methyl-1h-Pyrazol-3- Yl)Methyl]-N-Methylcarbamate | 1454848-24-8 |
Lurasidone | (1R,2R)-1,2-Cyclohexanedimethanol | 65376-05-8 |
Midazolam | 2-Amino-5-Chloro-2'-Fluorobenzophenone/BAT | 784-38-3 |
Mirogabalin | (1r,5s)-3-Ethyl-Bicyclo[3.2.0]Hept-3-En-6-One | 1235479-61-4 |
3-Ethylbicyclo[3.2.0]Hept-3-En-6-One | 1235479-59-0 | |
Tert-Butyl O,O-dimethylphosphonoacetate | 62327-21-3 | |
Montelukast sodium | A-[3-[2-(7-Chloro-2-Quinolinyl)Ethenyl]Phenyl]-2-(1-Hydroxy-1- Methylethyl)-,[S-(E)]-Benzenepropanol | 142569-70-8 |
2-[1-(Mercaptomethyl)Cyclopropyl]Acetic Acid | 162515-68-6 | |
Olmesartan | Ethyl 4-(1-Hydroxy-1-Methylethyl)-2-Propyl-Imidazole-5- Carboxylate/Imidazole Ester | 144689-93-0 |
DMDO-C1 | 80841-78-7 | |
Obeticholic Acid | Obeticholic Acid | 459789-99-2 |
(E)-3a-hydroxy-6-ethylidene-7-keto-5ẞ-cholan-24-oic acid | 1516887-33-4 | |
Rimegepant | 7,8-Dihydro-5H-Cyclohepta[b]pyridine-5,9(6H)-Dione | 39713-40-1 |
(R)-9-((Triisopropylsilyl)Oxy)-6,7,8,9-Tetrahydro-5h- Cyclohepta[b]Pyridin-5-Onehydrochloride Ester | 1190363-45-1 | |
(6S,9R)-6-(2,3-Difluorophenyl)-6,7,8,9-Tetrahydro-9-[[Tris(1- methylethyl)silyl]oxy]-5H-Cyclohepta[b]pyridin-5-One | 1190363-46-2 | |
Riociguat | 1-(2-Fluorobenzyl)-1h-Pyrazolo[3,4-B]Pyridine-3-Carbonitrile | 256376-65-5 |
Relugolix | 2-[2,6-Difluorobenzyl]Ethoxycarbonylamino]-4- [Dimethylaminomethyl]-5-4-Nitrophenylthiophene-3-Carboxylic acid | 1589503-95-6 |
Ethyl-2-Amino-4-Methyl-5-(4-Nitro-Phenyl) Thiophene-3- Carboxylate | 174072-89-0 | |
Ethyl 2-((2,6-difluorobenzyl)(ethoxycarbonyl)amino)-4-methyl-5-(4- nitrophenyl)thiophene-3-carboxylate | 308831-94-9 | |
Rocuronium bromide | (2b,3a,5a, 16b,17b)-2-(4-Morpholinyl)-16-(1-pyrrolidinyl)androstane3,17-diol LK-7 | 119302-20-4 |
Sacubitril | (2R,4S)-5-([1,1'-Biphenyl]-4-yl)-4-((Tert-Butoxycarbonyl)Amino)-2- Methylpentanoic Acid | 1012341-50-2 |
Sartans | 4-Methyl-2-Cyanobiphenyl (OTBN) | 114772-53-1 |
4'-Bromomethylbiphenyl-2-Carbonitrile (Br-OTBN) | 114772-54-2 | |
Sitagliptin | Sitagliptin Base | 486460-32-6 |
(2Z)-4-Oxo-4-[3-(Trifluoromethyl)-5,6-Dihydro-[1,2,4]Triazolo[4,3- A]Pyrazine-7(8H)-yl]-1-(2,4,5-Trifluorophenyl)Butan-2-One | 764667-65-4 | |
(R)-3-[(Tert-Butoxycarbonyl)amino]-4-(2,4,5-Trifluoro Phenyl)butanoic Acid | 486460-00-8 | |
Selpercatinib | 3,6-Diazabicyclo[3.1.1]heptane-6-carboxylic acid tert-butyl ester | 869494-16-6 |
4-(6-Fluoropyridin-3-Yl)-6-(2-Hydroxy-2- Methylpropoxy)Pyrazolo[1,5-A]Pyridine-3-Carbonitrile | 2222653-74-7 | |
4-(6-Fluoropyridin-3-yl)-6-hydroxурyrazolo[1,5-a]pyridine-3-carbonitrile | 2222654-09-1 | |
6-Bromo-4-Methoxурyrazolo[1,5-A]Pyridine-3-Carbonitrile | 1207836-10-9 | |
2-Fluoro-5-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-YI)Pyridine | 444120-95-0 | |
Semaglutide | tBuO-Ste-Glu(AEEA-AEEA-OH)-OtBu | 1118767-16-0 |
Octadecanedioic acid mono tert-butyl ester | 843666-40-0 | |
L-Glutamic acid-1-tert-butylester | 45120-30-7 | |
Boc-L-His(Trt)-OH | 32926-43-5 | |
8-Amino-3,6-dioxaoctanoicacid | 134978-97-5 | |
Suvorexant | 5-Methyl-2-(2h-1,2,3-Triazol-2-YI)Benzoic Acid | 956317-36-5 |
Trilaciclib Dihydrochloride | Spiro[cyclohexane-1,9'(6'H)-pyrazino[1',2':1,5]pyrrolo[2,3- d]pyrimidine]-7'(8'H)-carboxylic acid, 2'-(methylthio)-6'-охо-, 1,1- dimethylethyl esterN-4 | 2170746-99-1 |
Tofacitinib | 3-Bis(4-Methylbenzoyloxy)succinate) | 477600-71-8 |
4-Chloro-7H-pyrrolo[2,3-d]pyrimidine | 3680-69-1 | |
Ubrogepant | (S)-2'-Oxo-1',2',5,7-Tetrahydrospiro[Cyclopenta[B]Pyridine-6,3'- Pyrrolo[2,3-B]Pyridine]-3-Carboxylicacid | 1375541-21-1 |
Upadacitinib | N-[5-[(4-Methylphenyl)sulfonyl]-5H-Pyrrolo[2,3-b]pyrazin-2- yl]carbamic Acid Ethyl Ester | 1869118-24-0 |
(3R,4S)-3-(2-Bromoacetyl)-4-Ethyl-1-Pyrrolidinecarboxylic Acid Phenylmethyl Ester | 1428243-26-8 | |
Venetoclax | 1-((4'-Chloro-5,5-Dimethyl-3,4,5,6-Tetrahydro-[1,1'-biphenyl]-2- yl)methyl)piperazine dihydrochloride | 1628047-87-9 |
3-Nitro-4-((tetrahydro-2H-pyran-4- yl)methylamino)benzenesulfonamide | 1228779-96-1 | |
Methyl 2-((1H-pyrrolo[2,3-b]pyridin-5-yl)oxy)-4-fluorobenzoate | 1235865-75-4 | |
Vericiguat | 5-Fluoro-1-(2-Fluorobenzy1)-1h-Pyrazolo[3,4-B]Pyridine-3- Carbonitrile | 1350653-26-7 |
Vibegron | (Triphenylphosphoranylidene)Acetaldehyde | 2136-75-6 |
(4-Nitrobenzyl)Triphenylphosphonium Bromide | 2767-70-6 | |
(6S)-4,6,7,8-tetrahydro-4-oxo-Pyrrolo[1,2-a]pyriMidine-6-carboxylic acid | 1190392-22-3 | |
Vilanterol | 2-[2-(6-Bromohexyloxy)Ethoxymethyl]-1,3-Dichlorobenzene | 503070-57-3 |
(5r)-5-(2,2-Dimethyl-4h-1,3-Benzodioxin-6-YI)-1,3-Oxazolidin-2- One | 452339-73-0 | |
Vonoprazan | 2'-Fluoroacetophenone | 445-27-2 |
Voriconazole | 4-Chloro-6-ethyl-5-fluoropyrimidine | 137234-74-3 |
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